SCHEMBL5725809

SCHEMBL5725809

Cc1ccccc1C(CCCNC1CCCc2onc(O)c21)c1ccccc1C

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.35
SCD5 Q86SK9 2/20 0.33
NPC1 O15118 3/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5725812 1.00 DHODH (0.35) DHODHSCD5NPC1ALDH1A1LMNA
SCHEMBL5724732 0.97 DHODH (0.34) DHODHSCD5NPC1ALDH1A1LMNA
SCHEMBL5724892 0.86 HTR2A (0.36) DHODHSCD5NPC1ALDH1A1LMNA
SCHEMBL5726347 0.85 CHRM2 (0.32) DHODHNPC1LMNASMN1; SMN2GAA
SCHEMBL5726344 0.85 CHRM2 (0.32) DHODHNPC1LMNASMN1; SMN2GAA
SCHEMBL5725224 0.83 CHRM2 (0.32) NPC1LMNASMN1; SMN2GAAKMT2A
SCHEMBL5725148 0.80 SOS1 (0.40) DHODHSCD5NPC1ALDH1A1LMNA
SCHEMBL5726290 0.80 SCN5A (0.38) ALDH1A1KMT2AMEN1
SCHEMBL5724740 0.79 SLC6A1 (0.36) DHODHNPC1ALDH1A1RAB9AKMT2A
SCHEMBL5724739 0.79 KDM4E (0.34) NPC1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed