SCHEMBL5724914

SCHEMBL5724914

CCOc1noc2c1[C@H](NCCCC(c1ccc(F)cc1)c1ccc(F)cc1)CCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 1/20 0.35
CACNA1F O60840 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
DRD2 P14416 1/20 0.33
TACR2 P21452 1/20 0.33
DRD1 P21728 1/20 0.33
DRD5 P21918 1/20 0.33
HRH2 P25021 1/20 0.33
ADRA1D P25100 1/20 0.33
TACR1 P25103 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
ADRA1B P35368 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD3 P35462 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724638 0.91 HTR2A (0.35) HTR2AHTR2CHRH1MEN1KMT2A
SCHEMBL7977242 0.85 SOS1 (0.37) ADRA1DHTR2AHTR2CADRA1AHRH1
SCHEMBL5726290 0.83 SCN5A (0.38) SCN5AMEN1KMT2AVPS4BVCP
SCHEMBL5726294 0.83 SCN5A (0.38) SCN5AMEN1KMT2AVPS4BVCP
SCHEMBL5726344 0.83 CHRM2 (0.32) MEN1KMT2ACHRM2CHRM4CHRM5
SCHEMBL5726347 0.83 CHRM2 (0.32) MEN1KMT2ACHRM2CHRM4CHRM5
SCHEMBL5725224 0.80 CHRM2 (0.32) MEN1KMT2ACHRM2CHRM4CHRM5
SCHEMBL8790642 0.80 CHRM2 (0.32) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5724916 0.80 CHRM2 (0.32) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL7976983 0.74 KDM4E (0.45) HTR2AHTR2COPRK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed