SCHEMBL5727552

SCHEMBL5727552

CC(F)(Cc1cc(F)cc(C#N)c1)CC1CN(C(c2ccc(C#N)cc2)c2cccc(Br)c2)C1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.34
OPRD1 P41143 1/20 0.33
MGLL Q99685 1/20 0.32
MEN1 O00255 1/20 0.31
GLA P06280 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072255 0.92 MEN1 (0.37) OPRD1MGLLMEN1GLATSHR
SCHEMBL4684882 0.90 MEN1 (0.36) OPRD1MGLLMEN1GLATSHR
SCHEMBL5727486 0.88 MGLL (0.37) OPRD1MGLLMEN1GLATSHR
SCHEMBL5727699 0.86 CNR1 (0.38) MGLLMEN1GLATSHRKMT2A
SCHEMBL5727680 0.85 MGLL (0.41) MGLLMEN1GLATSHRKMT2A
SCHEMBL4787427 0.84 CNR1 (0.36) MGLLMEN1GLATSHRKMT2A
SCHEMBL5727485 0.83 TSHR (0.37) OPRD1MGLLMEN1GLATSHR
SCHEMBL4080122 0.82 CNR1 (0.40) MGLLMEN1GLATSHRKMT2A
SCHEMBL5727631 0.82 MEN1 (0.37) SLC6A9MGLLMEN1GLATSHR
SCHEMBL3481436 0.81 NOTUM (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636181-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2006-03-22 EP claimed
WO-2005000809-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2005-01-06 WO claimed