SCHEMBL5728253

SCHEMBL5728253

CC(NC(=O)c1ccc(I)cc1NS(=O)(=O)C1=CC=CN2SNC=C12)c1ccc(F)cc1F

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.33
SCN1A P35498 1/20 0.33
SCN1B Q07699 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
CCKAR P32238 1/20 0.32
CCKBR P32239 1/20 0.32
SLC22A2 O15244 2/20 0.31
GPR139 Q6DWJ6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3903821 1.00 NR1I2 (0.33) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL3907629 0.94 NR1I2 (0.33) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL3899480 0.91 GPR139 (0.34) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL1890458 0.91 CCKBR (0.33) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL3900169 0.91 CCR2 (0.37) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL3902491 0.90 KCNA5 (0.38)
SCHEMBL3899485 0.89 PDE2A (0.40) GPR139
SCHEMBL3901585 0.87 KCNA5 (0.38) NR1I2SCN1ASCN1BSCN5ASCN8A
SCHEMBL3903757 0.87 L3MBTL1 (0.38) CCKARCCKBR
SCHEMBL3902499 0.87 PDPK1 (0.32) SLC22A2GPR139

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675837-A2 BENZO [1,2,5] THIADIAZOLE COMPOUNDS AS CCK2 MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-07-05 EP disclosed
WO-2005012275-A2 BENZO [1, 2, 5] THIADIAZOLE COMPOUNDS AS CCK2 MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-02-10 WO disclosed