SCHEMBL5728563

SCHEMBL5728563

COC(=O)Oc1cc(-c2ccccc2)sc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.61
GAA P10253 5/20 0.61
ALDH1A1 P00352 4/20 0.61
HPGD P15428 4/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
ALOX15 P16050 8/20 0.52
IKBKB O14920 1/20 0.51
GFER P55789 1/20 0.51
TUBB4A P04350 2/20 0.51
TUBB P07437 2/20 0.51
TUBA3C P0DPH7 2/20 0.51
TUBA1B P68363 2/20 0.51
TUBA4A P68366 2/20 0.51
TUBB4B P68371 2/20 0.51
TUBB3 Q13509 2/20 0.51
TUBB2A Q13885 2/20 0.51
TUBB8 Q3ZCM7 2/20 0.51
TUBA3E Q6PEY2 2/20 0.51
TUBA1A Q71U36 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728244 0.86 IKBKB (0.56) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL27712944 0.85 MAPT (0.56) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL5728481 0.85 MAPT (0.50) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL5728267 0.85 ALDH1A1 (0.64) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL5727951 0.81 IKBKB (0.41) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL9409696 0.77 KDM4E (0.48) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL1563613 0.76 GAA (1.00) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL10639081 0.74 CYP1A1 (0.52) MAPTGAAALDH1A1HPGDMEN1
SCHEMBL5727996 0.74 JAK2 (0.40) ALDH1A1HPGDALOX15IKBKBTUBB4A
SCHEMBL5728140 0.73 HPGD (0.42) MAPTGAAALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694665-A2 SUBSTITUTED THIOPHENES AiCuris GmbH & Co. KG (DE) 2006-08-30 EP disclosed
WO-2006072348-A2 ALKINYL-SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2006-07-13 WO disclosed
WO-2005063734-A2 SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2005-07-14 WO disclosed