SCHEMBL5728643

SCHEMBL5728643

CC(=O)c1ccc(C)cc1C1CCCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.51
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
CAMKK2 Q96RR4 8/20 0.39
CAMKK1 Q8N5S9 3/20 0.39
OPRK1 P41145 1/20 0.39
KMT2A Q03164 2/20 0.39
GAA P10253 1/20 0.39
DDB1 Q16531 1/20 0.38
CRBN Q96SW2 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
KDM4E B2RXH2 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17682016 0.93 DRD2 (0.44) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL27652147 0.86 PTGDR2 (0.55) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL18304696 0.85 PTGDR2 (0.57) PTGDR2NPC1RAB9ACAMKK2CAMKK1
SCHEMBL27832665 0.82 PTGDR2 (0.51) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL4334283 0.81 PTGDR2 (0.47) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL9220646 0.81 PTGDR2 (0.50) PTGDR2NPC1RAB9AKMT2AGAA
SCHEMBL27832639 0.81 PTGDR2 (0.53) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL27436953 0.80 PTGDR2 (0.44) PTGDR2NPC1RAB9ADRD2DRD4
SCHEMBL23981527 0.80 CAMKK2 (0.41) PTGDR2NPC1RAB9ACAMKK2CAMKK1
SCHEMBL7534043 0.80 CHRNA1 (0.42) PTGDR2CAMKK2CAMKK1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed