SCHEMBL5729489

SCHEMBL5729489

CS(=O)(=O)c1ccc(-c2c[nH]c(OC(=O)Nc3ccc(Oc4cccnc4)cc3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PORCN Q9H237 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 2/20 0.43
PTGS2 P35354 2/20 0.43
HTT P42858 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
NAMPT P43490 6/20 0.41
SIRT6 Q8N6T7 1/20 0.40
PIP4K2A P48426 1/20 0.39
PIP4K2B P78356 1/20 0.39
NTRK1 P04629 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9106342 0.86 ALDH1A1 (0.51) PORCNSMN1; SMN2LMNAALDH1A1HTT
SCHEMBL4477095 0.86 ALDH1A1 (0.51) SMN1; SMN2LMNAALDH1A1PTGS2HTT
SCHEMBL9106921 0.81 HPGD (0.48) PORCNSMN1; SMN2LMNAALDH1A1NPC1
SCHEMBL9101092 0.79 KDR (0.49) PORCNSMN1; SMN2LMNAALDH1A1HTT
SCHEMBL9102775 0.75 SMN1; SMN2 (0.49) PORCNSMN1; SMN2LMNAALDH1A1HTT
SCHEMBL4473380 0.71 ALDH1A1 (0.57) SMN1; SMN2LMNAALDH1A1HTTTDP1
SCHEMBL9100139 0.69 KDR (0.60)
SCHEMBL5337025 0.68 ALDH1A1 (0.67) SMN1; SMN2LMNAALDH1A1HTTTDP1
SCHEMBL5725866 0.67 CDK8 (0.50) HTTGAARAB9A
SCHEMBL2645628 0.67 PTGS2 (0.50) SMN1; SMN2LMNAALDH1A1PTGS2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685125-B1 Pyrrole derivatives useful for the treatment of proliferative diseases MERCK PATENT GMBH (DE) 2012-06-06 EP disclosed
EP-1685125-A1 PYRROL DERIVATIVES MERCK PATENT GmbH (DE) 2006-08-02 EP disclosed
WO-2005049603-A1 PYRROL DERIVATIVES MERCK PATENT GMBH (DE) 2005-06-02 WO disclosed