SCHEMBL4477095

SCHEMBL4477095

CS(=O)(=O)c1ccc(-c2c[nH]c(C(=O)Nc3ccc(Oc4cccnc4)cc3)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
LMNA P02545 1/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
HTT P42858 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48
TP53 P04637 1/20 0.45
RECQL P46063 1/20 0.45
PTGS2 P35354 2/20 0.44
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
NAMPT P43490 2/20 0.42
HDAC3 O15379 1/20 0.41
BRAF P15056 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4473380 0.86 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5729489 0.86 PORCN (0.46) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL4475028 0.80 PGR (0.52) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL4477516 0.78 NPC1 (0.51) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL4472396 0.75 HTT (0.54) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL4465323 0.75 ROCK2 (0.50) NAMPT
SCHEMBL9106342 0.71 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL7302329 0.69 RAB9A (0.76) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL4466890 0.69 KDR (0.61) BRAFKDRCDK8
SCHEMBL4474468 0.69 KDR (0.46) NAMPTBRAFKDRCCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598274-B2 N-methyl-4-{4-[5-(4-chloro-3-trifluoromethylphenylcarbamoyl)-1H-pyrrol-3-yl]-phenoxy}pyridine-2-carboxamide; Raf kinases inhibitors MERCK PATENT GMBH (DE) 2009-10-06 US disclosed
US-20070149594-A1 Pyrrole derivatives MERCK PATENT GMBH (DE) 2007-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149594-A1 Pyrrole derivatives RAF1, BRAF, ARAF ALDH1A1 1625/4885SMN1; SMN2 4071/4885LMNA 2851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.