SCHEMBL5730481

SCHEMBL5730481

CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NNC(=O)OC(C)(C)C

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.67
CTSK P43235 4/20 0.67
CA2 P00918 1/20 0.52
KLK5 Q9Y337 1/20 0.47
KDM4E B2RXH2 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.46
HPGD P15428 2/20 0.45
LMNA P02545 1/20 0.45
THRB P10828 1/20 0.45
KLK7 P49862 1/20 0.44
EPHX2 P34913 1/20 0.44
BACE1 P56817 4/20 0.44
HSD17B10 Q99714 1/20 0.41
REN P00797 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL5730158 0.96 CTSS (0.63) CTSSCTSKCA2KLK5KDM4E
SCHEMBL1105463 0.87 CTSK (0.69) CTSSCTSKCA2KLK5KDM4E
SCHEMBL21887355 0.87 CTSK (0.69) CTSSCTSKCA2KLK5KDM4E
SCHEMBL1918995 0.87 CTSS (0.69) CTSSCTSKCA2KLK5KDM4E
SCHEMBL3757938 0.87 CTSS (0.69) CTSSCTSKCA2KLK5KDM4E
SCHEMBL1918997 0.87 CTSS (0.69) CTSSCTSKCA2KLK5KDM4E
SCHEMBL10210703 0.85 CTSS (0.67) CTSSCTSKCA2KLK5KDM4E
SCHEMBL18793329 0.85 CTSS (0.67) CTSSCTSKCA2KLK5KDM4E
SCHEMBL29147405 0.85 CTSS (0.67) CTSSCTSKCA2KLK5KDM4E
SCHEMBL15081482 0.83 CTSK (0.64) CTSSCTSKCA2KLK5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1188755-B1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-05-03 EP disclosed
US-6723722-B1 BLOOD COAGULATION FACTOR X INHIBITORS; ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-04-20 US disclosed
EP-1188755-A1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-20 EP disclosed