SCHEMBL5733736

SCHEMBL5733736

CCOC(=O)c1nc(-c2ccncc2)cs1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 10/20 0.53
DBF4 Q9UBU7 9/20 0.53
ALDH1A1 P00352 3/20 0.52
HPGD P15428 2/20 0.52
HSD17B10 Q99714 2/20 0.52
CASP1 P29466 1/20 0.51
CDK5 Q00535 5/20 0.49
CDK5R1 Q15078 5/20 0.49
MAPK1 P28482 1/20 0.47
CLK1 P49759 1/20 0.47
UBE2N P61088 1/20 0.47
ROCK2 O75116 1/20 0.46
PIM1 P11309 1/20 0.46
GSK3B P49841 1/20 0.46
HIPK2 Q9H2X6 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MMP2 P08253 1/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2705788 0.88 KDM4E (0.56) ALDH1A1HPGDMAPK1MEN1NPC1
SCHEMBL694852 0.88 ALDH1A1 (0.56) CDC7DBF4ALDH1A1HPGDHSD17B10
SCHEMBL28928759 0.87 ESR1 (0.49) ALDH1A1HPGDMAPK1MEN1NPC1
SCHEMBL10222539 0.86 ALDH1A1 (0.58) ALDH1A1HPGDHSD17B10MAPK1MMP13
SCHEMBL3612395 0.86 MAPT (0.57) ALDH1A1HPGDHSD17B10MAPK1MEN1
SCHEMBL1173463 0.86 PRKCZ (0.54) CDC7DBF4ALDH1A1HPGDHSD17B10
SCHEMBL204475 0.85 L3MBTL1 (0.57) ALDH1A1HPGDCDK5CDK5R1MAPK1
SCHEMBL4408696 0.85 KDM4E (0.59) ALDH1A1HPGDMEN1NPC1MAPT
SCHEMBL18425631 0.85 RAB9A (0.57) ALDH1A1MAPK1MEN1NPC1MAPT
SCHEMBL17396331 0.82 GAA (0.56) ALDH1A1HPGDMAPK1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986551-B1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA PHARMACEUTICAL (JP) 2006-08-02 EP disclosed
US-6359134-B1 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-19 US disclosed
EP-0986551-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Pharmaceutical Company Limited (JP) 2000-03-22 EP disclosed
WO-1998054164-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-03 WO disclosed