SCHEMBL5734401

SCHEMBL5734401

NC(=O)C1CCCN1C(=O)Nc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.63
RAB9A P51151 1/20 0.63
ALDH1A1 P00352 2/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
KMT2A Q03164 2/20 0.60
THRB P10828 1/20 0.60
ALOX12 P18054 1/20 0.60
FKBP1A P62942 2/20 0.59
KDM4E B2RXH2 1/20 0.57
HTT P42858 1/20 0.57
POLB P06746 1/20 0.55
ITGB3 P05106 1/20 0.54
ITGB1 P05556 1/20 0.54
ITGAV P06756 1/20 0.54
ITGA5 P08648 1/20 0.54
ITGA4 P13612 1/20 0.54
MTOR P42345 1/20 0.52
DPP4 P27487 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL10827466 0.99 NPC1 (0.62) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL1097863 0.96 NPC1 (0.62) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL4186674 0.88 KMT2A (0.76) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL27627515 0.87 ALDH1A1 (0.79) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL28721213 0.86 CCR1 (0.62) SMN1; SMN2KMT2ATHRBALOX12MTOR
SCHEMBL5735075 0.84 ALDH1A1 (0.74) SMN1; SMN2RAB9AALDH1A1CYP2C9KMT2A
SCHEMBL7309663 0.84 THRB (0.70) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL23418057 0.83 ALDH1A1 (0.70) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9
SCHEMBL31717915 0.82 CCR1 (0.59) CYP2C9CYP2C19KMT2ATHRBALOX12
SCHEMBL10364533 0.82 ITGB3 (0.58) NPC1SMN1; SMN2RAB9AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114591212-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2022-06-07 CN disclosed
CN-108289893-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2022-04-12 CN disclosed
EP-1268419-B1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-21 EP disclosed
EP-1268418-B1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-14 EP disclosed