SCHEMBL5734937

SCHEMBL5734937

COC(=O)C(C)(F)c1ccc2oc(CC(C)(C)C)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.45
AGPAT2 O15120 2/20 0.41
GAA P10253 1/20 0.39
AKR1B1 P15121 1/20 0.38
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
CETP P11597 1/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 1/20 0.36
UTRN P46939 1/20 0.36
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
MEN1 O00255 1/20 0.34
STAT3 P40763 1/20 0.34
KMT2A Q03164 1/20 0.34
SLC27A1 Q6PCB7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6785675 0.86 GAA (0.44) ACLYAGPAT2GAAAKR1B1HDAC3
SCHEMBL21130280 0.80 AKR1B1 (0.44) ACLYAGPAT2GAAAKR1B1HDAC3
SCHEMBL6790783 0.77 GAA (0.43) ACLYAGPAT2GAAAKR1B1HDAC3
SCHEMBL5736818 0.74 ACLY (0.39) ACLYAGPAT2GAAAKR1B1CETP
SCHEMBL28876443 0.73 NPC1 (0.46) ACLYGAAAKR1B1HDAC3HDAC1
SCHEMBL30358398 0.73 NPC1 (0.46) ACLYGAAAKR1B1HDAC3HDAC1
SCHEMBL5733868 0.73 NPC1 (0.45) ACLYGAARAB9ANPC1MAPT
SCHEMBL7978062 0.72 CA12 (0.48) ACLYGAARAB9ANPC1MEN1
SCHEMBL7997955 0.72 ACLY (0.42) ACLYRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL7997880 0.71 ESR1 (0.50) ACLYGAARAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1686128-A2 Isothiazole derivatives and their use as pesticides Syngenta Limited (GB) 2006-08-02 EP disclosed
EP-1265892-B1 ISOTHIAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES SYNGENTA LTD (GB) 2006-01-18 EP disclosed
US-6703347-B2 INSECTICIDES, FUNGICIDES, NEMATOCIDES, MOLLUSCICIDES, AND MITICIDES FOR PLANTS SYNGENTA LIMITED (GB) 2004-03-09 US disclosed
US-20030207926-A1 Isothiazole derivatives and their use as pesticides SYNGENTA LIMITED (GB) 2003-11-06 US disclosed
EP-1265892-A1 ISOTHIAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES Syngenta Limited (GB) 2002-12-18 EP disclosed
WO-2001055144-A1 ISOTHIAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES SYNGENTA LIMITED (GB) 2001-08-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030207926-A1 Isothiazole derivatives and their use as pesticides CBR1, CBR3, CYP1B1 ACLY 2189/4885AGPAT2 1916/4885GAA 4838/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.