SCHEMBL573693

SCHEMBL573693

COc1cc(N(C(=O)OC(C)(C)C)C2CCNCC2)ccc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 2/20 0.39
ALDH1A1 P00352 3/20 0.37
LMNA P02545 2/20 0.37
CHEK1 O14757 2/20 0.36
SIRT6 Q8N6T7 1/20 0.35
MAPT P10636 4/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A3 Q01959 1/20 0.35
TACR1 P25103 4/20 0.35
MAPK1 P28482 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
EHMT2 Q96KQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL573598 0.84 QPCT (0.41) QPCTALDH1A1SLC6A4SLC6A2SLC6A3
SCHEMBL574202 0.83 LMNA (0.36) ALDH1A1LMNAMAPTEHMT2
SCHEMBL4439400 0.82 POLB (0.40) ALDH1A1LMNAMAPTMAPK1KDM4E
SCHEMBL2578935 0.81 SLC6A4 (0.34) SLC6A4SLC6A2SLC6A3TACR1
SCHEMBL4436014 0.80 TACR1 (0.38) MAPTSLC6A4SLC6A2SLC6A3TACR1
SCHEMBL4434425 0.79 KDM4E (0.39) ALDH1A1LMNASLC6A4SLC6A2TACR1
SCHEMBL573664 0.78 SMN1; SMN2 (0.42) QPCTALDH1A1LMNACHEK1SIRT6
SCHEMBL4438391 0.78 KMT2A (0.36) ALDH1A1LMNAMAPTSLC6A4SLC6A2
SCHEMBL4433895 0.77 KDM4E (0.39) ALDH1A1LMNASLC6A4SLC6A2TACR1
SCHEMBL4444516 0.76 MAPK1 (0.40) ALDH1A1LMNAMAPTSLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601186-A2 4-(1H-INDOL-3-YL)-PYRIMIDINES AS ALK INHIBITORS AstraZeneca AB (SE) 2013-06-12 EP disclosed
WO-2012017239-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2012-02-09 WO disclosed