SCHEMBL5739199

SCHEMBL5739199

CS(=O)(=O)C1(S(C)(=O)=O)Oc2ccc(CNC(=O)C(F)(F)F)cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
KMT2A Q03164 4/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 2/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CHRNA7 P36544 1/20 0.35
CNR2 P34972 1/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
PDK2 Q15119 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506707 0.84 TSHR (0.40) TSHRKMT2ARAB9ASMN1; SMN2MEN1
SCHEMBL10277484 0.75 TSHR (0.40) TSHRKMT2ARAB9ASMN1; SMN2MEN1
SCHEMBL10227666 0.70 PDK2 (0.44) TSHRKMT2ARAB9ASMN1; SMN2MEN1
SCHEMBL15773718 0.64 ALDH1A1 (0.50) ALDH1A1CA1CA2CA7CA14
SCHEMBL22535940 0.64 ALDH1A1 (0.48) KMT2ASMN1; SMN2MEN1ALDH1A1POLB
SCHEMBL11946799 0.64 HTR7 (0.38) SMN1; SMN2ALDH1A1HPGD
SCHEMBL15013037 0.64 SMN1; SMN2 (0.56) KMT2ARAB9ASMN1; SMN2MEN1ALDH1A1
SCHEMBL7850276 0.64 RIPK1 (0.49) RAB9ASMN1; SMN2ALDH1A1HPGDLMNA
SCHEMBL16176470 0.62 CA1 (0.51) TSHRPOLBCA1CA2CA7
SCHEMBL8220431 0.62 MMP13 (0.55) RAB9ASMN1; SMN2ALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed