SCHEMBL5740494

SCHEMBL5740494

COC(=O)Oc1cn2ncnc(C3C(=O)Nc4cc(C(F)(F)F)ccc43)c2c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.35
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MET P08581 4/20 0.33
LMNA P02545 1/20 0.32
MAPK14 Q16539 1/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP1A2 P05177 1/20 0.31
STK10 O94804 1/20 0.31
MAP4K4 O95819 1/20 0.31
RET P07949 1/20 0.31
PDGFRB P09619 1/20 0.31
FGFR1 P11362 1/20 0.31
DDR1 Q08345 1/20 0.31
NUAK2 Q9H093 1/20 0.31
SLK Q9H2G2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049401 0.86 KDR (0.47) KDRMAPK14
SCHEMBL5740055 0.85 MAPT (0.35) KDRMAPTMETMAPK14
SCHEMBL5740281 0.85 CHEK1 (0.42) KDRMAPTTP53SMN1; SMN2MET
SCHEMBL5738802 0.85 KDR (0.32) KDRMAPTTP53METMAPK14
SCHEMBL5739596 0.83 MET (0.39) KDRMETMAPK14CYP3A4CYP2D6
SCHEMBL4111465 0.83 MAPK14 (0.36) KDRLMNAMAPK14
SCHEMBL5740803 0.81 MAPK14 (0.41) KDRMETMAPK14CYP3A4CYP2D6
SCHEMBL5740106 0.80 SYK (0.37) KDRMAPTTP53SMN1; SMN2MET
SCHEMBL5740319 0.80 KDR (0.37) KDRMETMAPK14CYP3A4CYP2D6
SCHEMBL5739297 0.79 MAPT (0.34) KDRMAPTTP53METLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed