SCHEMBL5740654

SCHEMBL5740654

COC(=O)c1cnccc1-c1ccc(C)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 1/20 0.64
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 2/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 2/20 0.46
ALPL P05186 1/20 0.46
POLB P06746 1/20 0.46
RAB9A P51151 1/20 0.46
SLC6A3 Q01959 3/20 0.45
SLC6A4 P31645 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SLC2A1 P11166 1/20 0.45
LMNA P02545 1/20 0.45
SLC22A12 Q96S37 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
TDP1 Q9NUW8 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29108469 0.89 CYP46A1 (0.65) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL30640092 0.89 CYP46A1 (0.65) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL5905310 0.86 SLC6A3 (0.63) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL6927417 0.86 FGFR1 (0.58) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL8217561 0.85 CASP1 (0.48) CYP46A1ALDH1A1KDM4EGAAMAPT
SCHEMBL1440123 0.80 SIRT3 (0.61) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL30957166 0.80 SIRT3 (0.61) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL23542701 0.80 SLC6A2 (0.56) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL14840639 0.78 CYP46A1 (1.00) CYP46A1ALDH1A1KDM4EGLAGAA
SCHEMBL11296276 0.78 KDM4E (0.51) CYP46A1ALDH1A1KDM4EGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678138-A1 PYRIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV Takeda Pharmaceutical Company Limited (JP) 2006-07-12 EP disclosed
WO-2005042488-A1 PYRIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-05-12 WO disclosed