SCHEMBL5740762

SCHEMBL5740762

COC(=O)Oc1cn2ncnc(C3C(=O)Nc4ccc(S(=O)(=O)N(C)C)cc43)c2c1C

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 4/20 0.31
TP53 P04637 2/20 0.31
POLB P06746 1/20 0.31
CHEK1 O14757 1/20 0.31
CDK1 P06493 1/20 0.31
CDK2 P24941 1/20 0.31
GSK3B P49841 1/20 0.31
ALDH1A1 P00352 4/20 0.30
MET P08581 2/20 0.30
KDM4E B2RXH2 2/20 0.30
GAA P10253 2/20 0.30
TTK P33981 1/20 0.30
HPGD P15428 1/20 0.30
THRB P10828 1/20 0.30
KDR P35968 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740106 0.91 SYK (0.37) KMT2AMEN1MAPTTP53ALDH1A1
SCHEMBL5739297 0.89 MAPT (0.34) MAPTTP53ALDH1A1METKDM4E
SCHEMBL14469831 0.87 MAPK14 (0.42) POLBKDR
SCHEMBL4053348 0.87 MAPK14 (0.42) POLBKDR
SCHEMBL5739782 0.86 MAPT (0.36) MAPTTP53POLBALDH1A1KDM4E
SCHEMBL5739596 0.85 MET (0.39) METKDRCYP3A4CYP2D6CYP2C9
SCHEMBL5740995 0.85 MET (0.33) METKDRCYP3A4
SCHEMBL5738334 0.85 KDM4E (0.43) MAPTTP53ALDH1A1KDM4E
SCHEMBL5738802 0.85 KDR (0.32) MAPTTP53METKDRCYP3A4
SCHEMBL5740803 0.85 MAPK14 (0.41) METKDRCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed