SCHEMBL5744301

SCHEMBL5744301

NN(C(=O)c1ccc(F)cc1)C(=O)[C@H]1CCCNC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
CYP2D6 P10635 1/20 0.43
SLC6A1 P30531 2/20 0.41
SLC6A11 P48066 1/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SLC6A13 Q9NSD5 1/20 0.41
NSD2 O96028 1/20 0.38
AGER Q15109 2/20 0.36
CDK9 P50750 2/20 0.36
NOS2 P35228 1/20 0.36
MTNR1A P48039 1/20 0.36
OPRD1 P41143 1/20 0.36
CHEK1 O14757 2/20 0.35
CDK2AP1 O14519 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5746273 1.00 KDM4E (0.43) KDM4EMAPTKMT2AATMCYP2D6
Hydrochloric Acid SCHEMBL5743267 0.99 KDM4E (0.42) KDM4EMAPTKMT2AATMCYP2D6
Hydrochloric Acid SCHEMBL5745261 0.99 KDM4E (0.42) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL2323451 0.79 HSD11B1 (0.49) KDM4EMAPTKMT2AATMCYP2D6
Hydrochloric Acid SCHEMBL5478791 0.77 HSD11B1 (0.48) KDM4EMAPTKMT2AATMCYP2D6
Hydrochloric Acid SCHEMBL192384 0.75 CDK9 (0.46) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL4678821 0.73 GLA (0.52) KDM4EKMT2AATMSMN1; SMN2ALDH1A1
SCHEMBL3879671 0.73 NPC1 (0.47) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL2597848 0.70 SLC6A1 (0.42) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL8110383 0.70 MEN1 (0.59) KDM4EKMT2ACYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685105-A1 ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2006-08-02 EP disclosed
WO-2005044797-A1 ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-05-19 WO disclosed