SCHEMBL3879671

SCHEMBL3879671

O=C(NC(=O)[C@H]1CCCNC1)c1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
KMT2A Q03164 2/20 0.45
KCNH2 Q12809 1/20 0.43
CDK9 P50750 1/20 0.43
SLC6A1 P30531 2/20 0.42
SLC6A11 P48066 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLC6A13 Q9NSD5 1/20 0.42
ALOX5 P09917 1/20 0.42
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3877272 0.85 TAS1R3 (0.45) CDK9SLC6A1SLC6A11TSHRLMNA
SCHEMBL6203700 0.83 KDM4E (0.45) KMT2ASLC6A1SLC6A11TSHRLMNA
SCHEMBL16333620 0.82 KMT2A (0.52) NPC1RAB9AKMT2AKCNH2ALOX5
SCHEMBL2323451 0.81 HSD11B1 (0.49) KMT2ASLC6A1SLC6A11TSHRLMNA
SCHEMBL2449552 0.80 ULK1 (0.56) NPC1RAB9AKMT2ACDK9
Hydrochloric Acid SCHEMBL5478791 0.80 HSD11B1 (0.48) KMT2ASLC6A1SLC6A11TSHRLMNA
SCHEMBL6203499 0.79 HDAC1 (0.48)
SCHEMBL6203532 0.79 HDAC1 (0.48)
SCHEMBL6204321 0.79 HDAC1 (0.48)
Hydrochloric Acid SCHEMBL193349 0.79 ULK1 (0.55) NPC1RAB9AKMT2ACDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2089386-A2 OXAZOLE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX Pharma S.A. (CH) 2009-08-19 EP disclosed
WO-2008056259-A2 OXAZOLE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMA S.A. (CH) 2008-05-15 WO disclosed