SCHEMBL5746358

SCHEMBL5746358

CCOC(c1ccc(-c2ccccc2N2CC(=O)ON2)cc1)c1nc2cccc(C(=O)O)c2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.34
ABCB11 O95342 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP2C9 P11712 1/20 0.34
ADRB3 P13945 1/20 0.34
ADRA2B P18089 1/20 0.34
SLC6A2 P23975 1/20 0.34
TBXAS1 P24557 1/20 0.34
HTR2C P28335 1/20 0.34
AGTR1 P30556 1/20 0.34
HTR2B P41595 1/20 0.34
AGTR2 P50052 1/20 0.34
PDE3A Q14432 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
MLKL Q8NB16 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789857 0.79 ABCB11 (0.36) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL844427 0.79 ABCB11 (0.38) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL6849453 0.74 AGTR1 (0.64) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL3638790 0.73 AGTR1 (0.39) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL9291479 0.71 PARP1 (0.35) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL8836872 0.71 BRS3 (0.33) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL3821755 0.70 AGTR2 (0.45) PPARGAGTR1AGTR2LTB4R2
SCHEMBL9638150 0.68 ABCB11 (0.37) PPARGABCB11EGFRERBB2CYP3A4
SCHEMBL4119807 0.67 DHODH (0.44)
SCHEMBL3400645 0.66 PPARG (0.51) PPARGCYP3A4ADORA3ADRA2BSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718641-A2 BENZIMIDAZOLE DERIVATIVE AND ITS USE AS AII RECEPTOR ANTAGONIST Takeda Pharmaceutical Company Limited (JP) 2006-11-08 EP disclosed
WO-2005080384-A2 BENZIMIDAZOLE DERIVATIVE AND USE AS AII RECEPTOR ANTAGONIST TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-09-01 WO disclosed