SCHEMBL5746771

SCHEMBL5746771

Fc1ccc2[c]ccc(F)c2c1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DAO P14920 1/20 0.31
CES2 O00748 2/20 0.30
CES1 P23141 2/20 0.30
MPO P05164 1/20 0.30
HTR2A P28223 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747398 0.83 CES2 (0.34) CA3CA6CA5ACA9CA14
SCHEMBL249073 0.73 CYP1A2 (0.31)
SCHEMBL27563254 0.71
SCHEMBL1448537 0.68 DAO (0.30) DAO
SCHEMBL5661873 0.67 LOXL2 (0.34)
SCHEMBL20356017 0.66 CA3 (0.48) CA3CA6CA5ACA9CA14
SCHEMBL7040909 0.65
SCHEMBL643603 0.65 CYP1A2 (0.48) ALDH1A1
SCHEMBL5660069 0.63 KCNQ3 (0.34)
SCHEMBL16585570 0.63 CYP1A2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901474-B1 ARYL PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-04-19 EP claimed
EP-0901474-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP claimed
US-5863924-A Aryl pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1999-01-26 US claimed
WO-1997044326-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-27 WO claimed
EP-1155698-A1 ORGANOBORON COMPOUNDS EXHIBITING ANTICOCCIDIAL ACTIVITIES Nitto Kasei Co., Ltd. (JP) 2001-11-21 EP disclosed