SCHEMBL5752285

SCHEMBL5752285

COc1ccc(CC(N)C(O)c2ccc(F)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
SLC6A4 P31645 1/20 0.50
FFAR1 O14842 1/20 0.47
LMNA P02545 2/20 0.47
MITF O75030 1/20 0.47
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
GPR35 Q9HC97 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
XBP1 P17861 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ATM Q13315 1/20 0.46
LDHA P00338 1/20 0.44
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749249 0.87 TRPA1 (0.47) HTTAOC3
SCHEMBL5751819 0.85 CYP2D6 (0.51) CYP1A2CYP2D6CYP2C19SLC6A4FFAR1
SCHEMBL5752240 0.83 TRPA1 (0.49) HTTMEN1KMT2AAOC3
SCHEMBL5751556 0.83 CASR (0.44) CYP1A2CYP2D6CYP2C19CNR1
SCHEMBL5750221 0.83 LTA4H (0.45) FFAR1
SCHEMBL5753279 0.81 TRPA1 (0.42) HTTAOC3
SCHEMBL7039221 0.81 CYP1A2 (0.83) CYP1A2CYP2D6CYP2C19SLC6A4FFAR1
SCHEMBL5749231 0.81 PTPN1 (0.39) CYP1A2CYP2D6CYP2C19CNR1
SCHEMBL5749180 0.79 LDHA (0.55) CYP1A2CYP2D6CYP2C19FFAR1LMNA
SCHEMBL5749784 0.78 TRPA1 (0.41) LMNAAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982348-B2 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-03 US disclosed
US-20040127574-A1 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-07-01 US disclosed
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127574-A1 Aminoethanol derivatives CETP, LCAT, MTTP CYP1A2 853/4885CYP2D6 1951/4885CYP2C19 1759/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.