SCHEMBL5749899

SCHEMBL5749899

CC(C)(C)c1ccc(CC(NC(=O)c2cccc3c(Cl)cccc23)C(OC(=O)CCC(=O)O)c2cccc(Cl)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.38
ADCY6 O43306 1/20 0.38
ADCY3 O60266 1/20 0.38
ADCY9 O60503 1/20 0.38
ADCY5 O95622 1/20 0.38
ADCY8 P40145 1/20 0.38
ADCY7 P51828 1/20 0.38
ADCY2 Q08462 1/20 0.38
ADCY1 Q08828 1/20 0.38
ADCY4 Q8NFM4 1/20 0.38
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
CNR1 P21554 2/20 0.34
CTSV O60911 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CNR2 P34972 1/20 0.34
MME P08473 4/20 0.34
NR1H4 Q96RI1 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579542 0.89 GCGR (0.35) GCGRADCY6ADCY3ADCY9ADCY5
SCHEMBL6579539 0.85 ITGB1 (0.35) GCGRADCY6ADCY3ADCY9ADCY5
SCHEMBL1897805 0.83 BACE1 (0.39) GCGRADCY6ADCY3ADCY9ADCY5
SCHEMBL5751437 0.82 ITGB1 (0.37) ITGB1ITGA4MMEPPARA
SCHEMBL5753208 0.78 ITGB1 (0.38) ITGB1ITGA4CNR2
SCHEMBL5751447 0.76 CTSV (0.36) ITGB1ITGA4CNR1CTSVCTSL
SCHEMBL5750208 0.76 CTSL (0.46) ITGB1ITGA4CTSVCTSLCTSB
SCHEMBL5751364 0.75 BACE1 (0.41) ITGB1ITGA4CTSVCTSLCTSB
SCHEMBL5752027 0.75 FFAR2 (0.37) ITGB1ITGA4CTSVCTSLCTSB
SCHEMBL5752124 0.75 BACE1 (0.38) CNR1CTSVCTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982348-B2 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-03 US disclosed