SCHEMBL575024

SCHEMBL575024

COC(NS(=O)(=O)c1cc(F)ccc1F)c1cccc(-c2ccnn2C2CCCCO2)c1F

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.39
CYP4A11 Q02928 3/20 0.39
ATR Q13535 14/20 0.39
ALPL P05186 2/20 0.35
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR7 P34969 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL574795 0.82 BRAF (0.39) ATRHTR1ADRD2HTR7HTR6
SCHEMBL574840 0.77 CYP4F2 (0.39) CYP4F2CYP4A11ATR
SCHEMBL575020 0.69 KDM1A (0.37) HTR1ADRD2HTR7HTR6
SCHEMBL574922 0.68 CYP4F2 (0.43) CYP4F2CYP4A11ATR
SCHEMBL22153397 0.67 ATR (0.40) CYP4F2CYP4A11ATR
SCHEMBL18536634 0.66 ATR (0.55) CYP4F2CYP4A11ATR
SCHEMBL574770 0.63 BRAF (0.37)
SCHEMBL15509064 0.62 CYP4F2 (0.47) CYP4F2CYP4A11ATR
SCHEMBL23535790 0.62 CYP4F2 (0.50) CYP4F2CYP4A11ATR
SCHEMBL24693881 0.62 CYP4F2 (0.50) CYP4F2CYP4A11ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601185-A1 DERIVATIVES OF PYRAZOLOPHENYL-BENZENESULFONAMIDE COMPOUNDS AND USE THEREOF AS ANTITUMOR AGENTS Nerviano Medical Sciences S.r.l. (IT) 2013-06-12 EP disclosed
WO-2012016993-A1 DERIVATIVES OF PYRAZOLOPHENYL-BENZENESULFONAMIDE COMPOUNDS AND USE THEREOF AS ANTITUMOR AGENTS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-02-09 WO disclosed