SCHEMBL5755875

SCHEMBL5755875

CCCCc1ccc(N(Br)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
RARB P10826 1/20 0.41
PLK1 P53350 1/20 0.41
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
FAAH O00519 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GALR3 O60755 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PLA2G1B P04054 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754826 0.80 PPARA (0.48) HDAC3HDAC1HDAC2NCOR2
SCHEMBL177445 0.79 THRA (0.47) ALDH1A1HSD17B10RARBTHRATHRB
SCHEMBL1007329 0.77 MT-CO2 (0.51) ALDH1A1POLB
SCHEMBL1008034 0.77 MT-CO2 (0.39) HPGDALDH1A1RAB9AKDM4E
SCHEMBL3332104 0.76 HPGD (0.43) HPGDALDH1A1HSD17B10NPC1RAB9A
SCHEMBL5756917 0.75 HDAC3 (0.37) THRATHRBHDAC3HDAC1HDAC2
SCHEMBL7112682 0.75 KCNH2 (0.41) ALDH1A1RARBTHRATHRBFAAH
SCHEMBL3339006 0.74 HPGD (0.41) HPGDALDH1A1HSD17B10NPC1RAB9A
SCHEMBL6404151 0.72 CYP4A11 (0.46) HPGDALDH1A1HSD17B10CA2
SCHEMBL6405545 0.72 CYP4Z1 (0.41) HPGDALDH1A1HSD17B10THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP disclosed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP disclosed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO disclosed