SCHEMBL5758045

SCHEMBL5758045

O=CNCCC(c1ccccc1)N1CCC(C(=O)c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
CCR3 P51677 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42
KCNH2 Q12809 1/20 0.42
SCD O00767 1/20 0.41
CPB1 P15086 1/20 0.41
KMT2A Q03164 3/20 0.41
MGLL Q99685 2/20 0.41
MEN1 O00255 2/20 0.41
HSD11B1 P28845 1/20 0.41
SLC18A3 Q16572 1/20 0.40
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
PRSS1 P07477 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754847 0.86 EPHX2 (0.53) HTR2ACCR3CYP1A2CYP2C9HPGD
SCHEMBL5757058 0.82 SLC18A3 (0.47) HTR2ACCR3MGLLSLC18A3
Hydrochloric Acid SCHEMBL5755104 0.81 HTR2A (0.47) HTR2ACCR3CYP1A2CYP2C9HPGD
SCHEMBL5756913 0.80 CYP2C19 (0.51) CYP1A2CYP2C9CYP2C19HSD11B1
SCHEMBL5755428 0.80 SLC6A2 (0.47) HTR2ACCR3CYP1A2KCNH2KMT2A
SCHEMBL5758947 0.76 SIGMAR1 (0.46) CCR3KCNH2KMT2AMEN1
SCHEMBL5757158 0.75 HSD11B1 (0.54) HTR2ACYP1A2HSD11B1
SCHEMBL9377800 0.73 HSD11B1 (0.57) HTR2ACYP1A2HSD11B1
SCHEMBL6007500 0.73 HTR2A (0.55) HTR2ACCR3CYP1A2KCNH2
SCHEMBL27298639 0.71 HTR2A (0.56) HTR2ACCR3KCNH2CPB1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP claimed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP claimed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO claimed
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP disclosed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP disclosed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO disclosed