SCHEMBL5759683

SCHEMBL5759683

c1ccc(COc2ccc(COc3ccc(CCCn4ccnc4)cc3)cn2)cc1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 2/20 0.71
QPCT Q16769 1/20 0.54
LTA4H P09960 1/20 0.53
KMT2A Q03164 1/20 0.52
CYP19A1 P11511 2/20 0.51
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
TBXAS1 P24557 3/20 0.48
CACNA1B Q00975 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5759785 0.91 HMOX1 (0.85) HMOX1QPCTLTA4HKMT2ACYP19A1
SCHEMBL5757778 0.87 HMOX1 (0.83) HMOX1QPCTLTA4HKMT2ACYP19A1
SCHEMBL5760109 0.79 HMOX1 (0.65) HMOX1QPCTKMT2ACYP19A1TBXAS1
SCHEMBL3160306 0.78 CYP19A1 (0.71) HMOX1QPCTCYP19A1CYP11B1CYP11B2
SCHEMBL5759974 0.77 HMOX1 (0.62) HMOX1QPCTLTA4HKMT2ACYP19A1
SCHEMBL5761690 0.77 HMOX1 (0.56) HMOX1QPCTLTA4HKMT2A
Hydrochloric Acid SCHEMBL411704 0.77 CYP19A1 (0.69) HMOX1QPCTCYP19A1CYP11B1CYP11B2
SCHEMBL5759151 0.76 HMOX1 (0.64) HMOX1QPCTKMT2ACYP19A1
SCHEMBL7477480 0.76 HMOX1 (0.75) HMOX1QPCTLTA4HKMT2ACYP19A1
SCHEMBL5760287 0.75 CYP11B1 (0.59) HMOX1KMT2ACYP19A1CYP11B1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed