SCHEMBL5761774

SCHEMBL5761774

CS(=O)(=O)N(Cc1ccccc1)c1ncc(Br)cn1.[NaH]

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
L3MBTL1 Q9Y468 2/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
GAA P10253 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
PTPN11 Q06124 1/20 0.38
POLB P06746 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.37
GBA1 P04062 1/20 0.37
NR1I2 O75469 1/20 0.37
APOBEC3A P31941 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2114576 0.98 ALDH1A1 (0.56) ALDH1A1L3MBTL1TSHRHTTGAA
SCHEMBL5761769 0.96 ALDH1A1 (0.54) ALDH1A1L3MBTL1TSHRHTTGAA
SCHEMBL2112891 0.85 GRM2 (0.47) ALDH1A1L3MBTL1TSHRHTTSMN1; SMN2
SCHEMBL20394335 0.74 LMNA (0.48) ALDH1A1TSHRHTTSMN1; SMN2GBA1
SCHEMBL12808838 0.72 ALDH1A1 (0.60) ALDH1A1L3MBTL1TSHRHTTGAA
SCHEMBL2111862 0.72 TSPO (0.50) ALDH1A1L3MBTL1TSHRGAASMN1; SMN2
SCHEMBL2113204 0.72 ALDH1A1 (0.43) ALDH1A1HTTGAASMN1; SMN2MEN1
SCHEMBL7095387 0.69 ALDH1A1 (0.60) ALDH1A1GAASMN1; SMN2MEN1KMT2A
SCHEMBL5762013 0.69 EDNRA (0.33) ALDH1A1
SCHEMBL18438489 0.68 ALDH1A1 (0.62) ALDH1A1GAASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611091-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2006-01-04 EP disclosed
WO-2004089885-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-10-21 WO disclosed