SCHEMBL5763615

SCHEMBL5763615

COc1ccc2c(c1)C(=O)c1cc(NC(=O)C(C)(O)C(F)(F)F)ccc1CO2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 5/20 0.54
PDK2 Q15119 5/20 0.54
PDK3 Q15120 5/20 0.54
PDK4 Q16654 5/20 0.54
ALDH1A1 P00352 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
MAPT P10636 3/20 0.54
KDM4E B2RXH2 1/20 0.54
NPC1 O15118 1/20 0.54
GAA P10253 1/20 0.54
HPGD P15428 1/20 0.54
ALOX12 P18054 1/20 0.54
RAB9A P51151 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
MAPK14 Q16539 3/20 0.48
ABCC9 O60706 5/20 0.48
ABCC8 Q09428 5/20 0.48
KCNJ11 Q14654 5/20 0.48
KCNJ8 Q15842 5/20 0.48
PPIA P62937 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833166 0.86 ABCC9 (0.54) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL5766461 0.84 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2MAPTKDM4ENPC1
SCHEMBL87317 0.78 ALDH1A1 (0.83) ALDH1A1SMN1; SMN2MAPTKDM4ENPC1
SCHEMBL7829727 0.78 ABCC9 (0.44) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL7829722 0.78 ABCC9 (0.44) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL7832140 0.78 MAPK14 (0.56) PDK1PDK2PDK3PDK4MAPK14
SCHEMBL7833285 0.76 ABCC9 (0.49) PDK1PDK2PDK3PDK4MAPK14
SCHEMBL7829732 0.75 ABCC9 (0.58) PDK1PDK2PDK3PDK4ABCC9
SCHEMBL8796551 0.74 PDK1 (0.47) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL5766822 0.72 ALDH1A1 (0.71) ALDH1A1SMN1; SMN2MAPTKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979821-B1 TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO KK (JP) 2006-09-13 EP disclosed
US-6211227-B1 SULFUR CONTAINING TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-04-03 US disclosed
EP-0979821-A1 TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO CO., LTD. (JP) 2000-02-16 EP disclosed