SCHEMBL5764000

SCHEMBL5764000

COc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 15/20 1.00
EGFR P00533 9/20 1.00
SRC P12931 9/20 1.00
PDGFRB P09619 6/20 0.82
PDGFRA P16234 6/20 0.82
ABL1 P00519 5/20 0.80
MAPK14 Q16539 5/20 0.80
WEE1 P30291 3/20 0.79
FGFR2 P21802 1/20 0.79
FGFR4 P22455 1/20 0.79
FGFR3 P22607 1/20 0.79
KIT P10721 3/20 0.78
PSEN1 P49768 1/20 0.75
PSEN2 P49810 1/20 0.75
APH1B Q8WW43 1/20 0.75
NCSTN Q92542 1/20 0.75
APH1A Q96BI3 1/20 0.75
PSENEN Q9NZ42 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763930 0.92 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764023 0.91 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL1335649 0.90 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764062 0.90 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5762228 0.89 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5762046 0.89 SRC (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL1249524 0.89 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL10102543 0.89 FGFR1 (0.86) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL26257902 0.88 FGFR1 (0.79) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL1334768 0.88 SRC (1.00) FGFR1EGFRSRCPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP claimed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO claimed
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP disclosed