SCHEMBL5763930

SCHEMBL5763930

COc1cc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 16/20 1.00
EGFR P00533 13/20 1.00
SRC P12931 11/20 0.85
WEE1 P30291 2/20 0.76
FGFR2 P21802 1/20 0.76
FGFR4 P22455 1/20 0.76
FGFR3 P22607 1/20 0.76
PDGFRB P09619 8/20 0.75
PDGFRA P16234 8/20 0.75
ABL1 P00519 7/20 0.75
MAPK14 Q16539 7/20 0.75
KIT P10721 3/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764023 0.93 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5764000 0.92 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5762228 0.89 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL1249524 0.86 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL26257902 0.86 FGFR1 (0.79) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5762573 0.86 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL1334768 0.86 SRC (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5764062 0.85 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5764012 0.85 FGFR1 (1.00) FGFR1EGFRSRCWEE1FGFR2
SCHEMBL5762046 0.85 SRC (1.00) FGFR1EGFRSRCWEE1FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO claimed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP claimed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO claimed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO disclosed