SCHEMBL5762228

SCHEMBL5762228

COc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 14/20 1.00
EGFR P00533 11/20 1.00
SRC P12931 10/20 0.80
PDGFRB P09619 7/20 0.77
PDGFRA P16234 7/20 0.77
ABL1 P00519 6/20 0.77
MAPK14 Q16539 6/20 0.77
KIT P10721 3/20 0.77
WEE1 P30291 2/20 0.75
FGFR2 P21802 1/20 0.74
FGFR4 P22455 1/20 0.74
FGFR3 P22607 1/20 0.74
PSEN1 P49768 1/20 0.71
PSEN2 P49810 1/20 0.71
APH1B Q8WW43 1/20 0.71
NCSTN Q92542 1/20 0.71
APH1A Q96BI3 1/20 0.71
PSENEN Q9NZ42 1/20 0.71
RIPK2 O43353 1/20 0.70
ACVR1 Q04771 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763930 0.89 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764000 0.89 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764023 0.88 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL1334768 0.87 SRC (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764062 0.87 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL25399961 0.86 FGFR1 (0.82) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL30618363 0.86 FGFR1 (0.82) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5762046 0.86 SRC (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL5764012 0.86 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA
SCHEMBL1249524 0.86 FGFR1 (1.00) FGFR1EGFRSRCPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP claimed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO claimed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP claimed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO claimed
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP disclosed
WO-2005105097-A2 PYRIDOPYRIMIDINES FOR TREATING INFLAMMATORY AND OTHER DISEASES GPC BIOTECH AG (DE) 2005-11-10 WO disclosed