SCHEMBL576412

SCHEMBL576412

C=CCC1CCCOC1=O

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 2/20 0.41
CTRC Q99895 2/20 0.41
F2 P00734 1/20 0.41
NOS1 P29475 2/20 0.40
NOS2 P35228 2/20 0.40
FAAH O00519 1/20 0.33
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
FKBP1A P62942 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22643587 1.00 PRSS1 (0.41) PRSS1CTRCF2NOS1NOS2
SCHEMBL577127 0.94 NOS1 (0.42) PRSS1CTRCF2NOS1NOS2
SCHEMBL576860 0.88
SCHEMBL11915557 0.82 KCNH3 (0.31)
SCHEMBL10431427 0.81 FAAH (0.38) PRSS1CTRCF2FAAH
SCHEMBL27706139 0.80 PRSS1 (0.35) PRSS1CTRCF2
Acetic Acid SCHEMBL11034851 0.79 FAAH (0.36) PRSS1CTRCF2FAAH
SCHEMBL5013295 0.79 FAAH (0.41) PRSS1CTRCF2FAAH
SCHEMBL20980149 0.78 NOS1 (0.41) PRSS1CTRCF2NOS1NOS2
SCHEMBL24829919 0.78 NOS2 (0.33) NOS1NOS2FKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 192 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240368351-A1 FACTORS CONTROLLING DRUG RELEASE IN CROSS-LINKED POLY(VALEROLACTONE) BASED MATRICES PENDANT BIOSCIENCES INC (US) 2024-11-07 US claimed
US-11905377-B2 Factors controlling drug release in cross-linked poly(valerolactone) based matrices PENDANT BIOSCIENCES, INC. (US) 2024-02-20 US claimed
US-20140371403-A1 STENT FORMED FROM CROSSLINKED BIOABSORBABLE POLYMER ABBOTT CARDIOVASCULAR SYSTEMS (US) 2014-12-18 US claimed
US-8679396-B2 Method of making a stent formed from crosslinked bioabsorbable polymer ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2014-03-25 US claimed
US-20120149850-A1 STENT FORMED FROM CROSSLINKED BIOABSORBABLE POLYMER ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2012-06-14 US claimed
US-20120150283-A1 METHOD OF MAKING A STENT FORMED FROM CROSSLINKED BIOABSORBABLE POLYMER ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2012-06-14 US claimed
US-8147744-B2 Method of making a stent formed from crosslinked bioabsorbable polymer ABBOTT CARDIOVASCULAR SYSTEMS INC. (US) 2012-04-03 US claimed
EP-2266967-A1 Intermediates for the preparation of octahydroquinolizines 55pharma Drug Discovery & Development AG (AT) 2010-12-29 EP claimed
WO-2010144937-A2 INTERMEDIATES FOR THE PREPARATION OF OCTAHYDROQUINOLIZINES 55PHARMA DRUG DISCOVERY & DEVELOPMENT AG (AT) 2010-12-23 WO claimed
US-20100262223-A1 Stent Formed from Crosslinked Bioabsorbable Polymer and Methods of Making the Stent ABBOTT CARDIOVASCULAR SYSTEMS INC. 2010-10-14 US claimed
US-6346599-B1 CONDENSATION POLYMERIZATION OF LACTONE MIXTURE WITH INHIBITION OF CRYSTALLIZATION UNION CARBIDE CHEMICALS & PLASTICS TECHNOLOGY CORPORATION 2002-02-12 US claimed
EP-0559789-A1 PROCESS FOR THE PREPARATION OF $g(a)-ALKYL LACTONES HENKEL CORPORATION (US) 1993-09-15 EP claimed
WO-1992009590-A1 PROCESS FOR THE PREPARATION OF α-ALKYL LACTONES HENKEL CORPORATION (US) 1992-06-11 WO claimed
US-20240368351-A1 FACTORS CONTROLLING DRUG RELEASE IN CROSS-LINKED POLY(VALEROLACTONE) BASED MATRICES PENDANT BIOSCIENCES INC (US) 2024-11-07 US disclosed
US-20240368351-A1 FACTORS CONTROLLING DRUG RELEASE IN CROSS-LINKED POLY(VALEROLACTONE) BASED MATRICES PENDANT BIOSCIENCES INC (US) 2024-11-07 US disclosed
US-11905377-B2 Factors controlling drug release in cross-linked poly(valerolactone) based matrices PENDANT BIOSCIENCES, INC. (US) 2024-02-20 US disclosed
EP-0024682-B1 PROCESS FOR THE PREPARATION OF N-PROPYL-N-PROPYLIDENE ACETAMIDE OR DI-N-PROPYL ACETAMIDE Consortium für elektrochemische Industrie GmbH (DE) 1982-12-22 EP disclosed
EP-0003846-B1 A PROCESS FOR PRODUCING A CROSSLINKABLE COPOLYMER OF A LACTONE AND A POLYFUNCTIONAL ACRYLATE, THE SO OBTAINED COPOLYMER, A METHOD FOR THE MANUFACTURE OF ARTICLES THEREFROM AND THE SO FORMED ARTICLES UNION CARBIDE CORPORATION (US) 1982-10-20 EP disclosed
US-4315011-A VASODILATORS RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1982-02-09 US disclosed
EP-0024682-A1 Process for the preparation of n-propyl-n-propylidene acetamide or di-n-propyl acetamide Consortium für elektrochemische Industrie GmbH (DE) 1981-03-11 EP disclosed