SCHEMBL5765110

SCHEMBL5765110

CCc1cc2c(=O)nc[nH]c2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.37
CYP1A2 P05177 1/20 0.37
TMIGD3 P0DMS9 1/20 0.37
CYP2C9 P11712 1/20 0.37
ADORA1 P30542 1/20 0.37
DAO P14920 1/20 0.32
PDE4A P27815 2/20 0.31
ADORA2A P29274 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
KDM5B Q9UGL1 1/20 0.31
IP6K1 Q92551 1/20 0.31
CHEK1 O14757 2/20 0.30
PIM1 P11309 2/20 0.30
AKT1 P31749 1/20 0.30
FLT3 P36888 1/20 0.30
PIM3 Q86V86 1/20 0.30
RPS6KA3 P51812 1/20 0.30
ACVR1 Q04771 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410480 0.77 ADORA1 (0.38) PARP1CYP1A2ADORA1ADORA2AIP6K1
SCHEMBL13627444 0.73 PARP1 (0.36) PARP1IP6K1CHEK1PIM1AKT1
SCHEMBL5763588 0.72 PARP1 (0.37) PARP1ADORA1DAOADORA2A
SCHEMBL5765249 0.69 HTT (0.41) PARP1
SCHEMBL22283252 0.67 PDE3B (0.46) PARP1ADORA1CHEK1PIM1AKT1
SCHEMBL12410487 0.64 LMNA (0.50) CYP1A2KDM5BCHEK1
SCHEMBL26754441 0.62 GABRR1 (0.41) CYP1A2TMIGD3CYP2C9ADORA1PDE4A
SCHEMBL15707647 0.62 GSK3B (0.41) PARP1KDM5BCHEK1PIM1AKT1
SCHEMBL9134716 0.61 DAO (0.44) PARP1DAO
SCHEMBL1507437 0.61 ALDH1A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091738-B1 BICYCLIC sPLA 2 INHIBITORS LILLY CO ELI (US) 2006-12-06 EP disclosed
US-6384041-B1 ANTIINFLAMMATORY AGENT, TREATMENT OF SHOCK AND ENZYME INHIBITORS ELI LILLY AND COMPANY 2002-05-07 US disclosed