SCHEMBL5767550

SCHEMBL5767550

CC(C)S(=O)(=O)n1c(NCC2CC2)nc2ccc(C=N)cc21

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.38
PI4KB Q9UBF8 1/20 0.33
CNR2 P34972 1/20 0.32
CYP3A4 P08684 8/20 0.32
MET P08581 1/20 0.32
S1PR1 P21453 1/20 0.31
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774393 0.82 MAPK14 (0.38) MAPK14PI4KBCYP3A4
SCHEMBL5769574 0.81 PI4KB (0.36) MAPK14PI4KBCYP3A4
SCHEMBL5774512 0.80 ALDH1A1 (0.40) MAPK14PI4KBS1PR1
SCHEMBL5771593 0.80 PDE4B (0.37) MAPK14PI4KBCYP3A4
SCHEMBL5772303 0.80 PDE4B (0.37) MAPK14PI4KBCYP3A4
SCHEMBL5773723 0.80 MAPK14 (0.41) MAPK14CYP3A4
SCHEMBL5768603 0.79 FGFR2 (0.32) MAPK14PI4KBCNR2CYP3A4
SCHEMBL5768943 0.78 ALDH1A1 (0.47) MAPK14
SCHEMBL5770367 0.78 MAPK14 (0.41) MAPK14PI4KBCYP3A4
SCHEMBL5770827 0.78 TP53 (0.48) MAPK14PI4KBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-B1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE LILLY CO ELI (US) 2006-10-25 EP disclosed