SCHEMBL5773723

SCHEMBL5773723

CC(C)S(=O)(=O)n1c(NCc2ccc(F)cc2)nc2ccc(C=N)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.41
CYP3A4 P08684 8/20 0.39
RXFP1 Q9HBX9 1/20 0.38
GAA P10253 2/20 0.37
MAPT P10636 1/20 0.37
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
FYN P06241 1/20 0.36
PIM1 P11309 1/20 0.36
FGFR1 P11362 1/20 0.36
MAPK1 P28482 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
CSNK1D P48730 1/20 0.36
LIMK1 P53667 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDC42BPA Q5VT25 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5773725 0.89 MAPK14 (0.42) MAPK14CYP3A4GAAMAPTMAPK1
SCHEMBL5774512 0.89 ALDH1A1 (0.40) MAPK14GAAMAPTMAPK1KDM4E
SCHEMBL5770827 0.84 TP53 (0.48) MAPK14CYP3A4GAAMAPTMEN1
SCHEMBL5773732 0.83 KDM4E (0.38) MAPK14CYP3A4RXFP1GAAMAPT
SCHEMBL5774393 0.81 MAPK14 (0.38) MAPK14CYP3A4
SCHEMBL5768943 0.80 ALDH1A1 (0.47) MAPK14GAAMAPTKDM4EMEN1
SCHEMBL5767550 0.80 MAPK14 (0.38) MAPK14CYP3A4
SCHEMBL5769574 0.80 PI4KB (0.36) MAPK14CYP3A4
SCHEMBL5770367 0.78 MAPK14 (0.41) MAPK14CYP3A4GAAMEN1CYP2D6
SCHEMBL18058953 0.75 THRB (0.50) MAPK14CYP3A4RXFP1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-B1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE LILLY CO ELI (US) 2006-10-25 EP disclosed