SCHEMBL5770367

SCHEMBL5770367

CC(C)S(=O)(=O)n1c(NCCCc2ccccc2)nc2ccc(C=N)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.41
PI4KB Q9UBF8 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 1/20 0.35
KMT2A Q03164 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP3A4 P08684 2/20 0.35
POLB P06746 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3R1 P27986 1/20 0.34
GAA P10253 1/20 0.34
SLC2A1 P11166 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5773725 0.80 MAPK14 (0.42) MAPK14CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL5773732 0.80 KDM4E (0.38) MAPK14KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL5774512 0.79 ALDH1A1 (0.40) MAPK14PI4KBKMT2ACYP2C19GAA
SCHEMBL5770827 0.79 TP53 (0.48) MAPK14PI4KBKMT2ACYP2D6CYP2C9
SCHEMBL5773723 0.78 MAPK14 (0.41) MAPK14KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL5767550 0.78 MAPK14 (0.38) MAPK14PI4KBCYP3A4
SCHEMBL5769574 0.78 PI4KB (0.36) MAPK14PI4KBCYP3A4
SCHEMBL5772161 0.77 PI4KB (0.39) MAPK14PI4KBKMT2ACYP2C9CYP2C19
SCHEMBL5771480 0.77 SSTR5 (0.47) KMT2ALMNAHTTMEN1
SCHEMBL18058953 0.73 THRB (0.50) MAPK14PI4KBKMT2ACYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-B1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE LILLY CO ELI (US) 2006-10-25 EP disclosed