SCHEMBL5769284

SCHEMBL5769284

CC(C)(C)OC(=O)N1CCCCC1CCNc1ncc(Cl)c(CCOS(C)(=O)=O)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.40
TRPV1 Q8NER1 2/20 0.39
ATM Q13315 2/20 0.37
APP P05067 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
DRD2 P14416 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
SLC6A2 P23975 1/20 0.36
HRH2 P25021 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
DRD3 P35462 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
PSEN1 P49768 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515983 0.89 CHEK2 (0.40) CHEK2TRPV1ATMPRMT5PDE7B
SCHEMBL5801498 0.83 TRPV1 (0.41) CHEK2TRPV1ATMAPPHTR1A
SCHEMBL5773134 0.83 ATM (0.39) CHEK2TRPV1ATMPRMT5PDE7B
SCHEMBL5769599 0.79 ATM (0.38) CHEK2TRPV1ATMPRMT5PDE7B
SCHEMBL5479174 0.78 ATM (0.39) CHEK2TRPV1ATMAPPHTR1A
SCHEMBL5774380 0.78 ALDH1A1 (0.39) CHEK2TRPV1PRMT5PDE7BALDH1A1
SCHEMBL8262110 0.76 TRPV1 (0.40) CHEK2TRPV1ATMAPPHTR1A
SCHEMBL6174216 0.75 ATM (0.46) CHEK2TRPV1ATMAPPHTR1A
SCHEMBL2915181 0.75 ATM (0.46) CHEK2TRPV1ATMAPPHTR1A
SCHEMBL3126719 0.75 ATM (0.46) CHEK2TRPV1ATMAPPHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066899-A1 NOVEL THROMBIN INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) AG (CH) 2006-06-29 WO disclosed
EP-1674464-A1 Novel thrombin inhibitors Santhera Pharmaceuticals (Schweiz) GmbH (CH) 2006-06-28 EP disclosed
EP-1674464-A1 Novel thrombin inhibitors Santhera Pharmaceuticals (Schweiz) GmbH (CH) 2006-06-28 EP disclosed