SCHEMBL5774380

SCHEMBL5774380

CC(C)(C)OC(=O)N1CCCCC1CCNc1ncc(Cl)c(CCNCc2n[nH]c3ccc(Cl)cc23)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CHEK2 O96017 2/20 0.39
CNR1 P21554 2/20 0.38
PDE7B Q9NP56 1/20 0.37
PRMT5 O14744 1/20 0.36
CCNT1 O60563 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
AHCY P23526 1/20 0.33
METTL3 Q86U44 1/20 0.33
CHEK1 O14757 1/20 0.33
IKBKB O14920 1/20 0.33
AURKA O14965 1/20 0.33
PAK4 O96013 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5800853 0.87 ALDH1A1 (0.39) ALDH1A1CHEK2CNR1PDE7BPRMT5
SCHEMBL5479053 0.82 ALDH1A1 (0.37) ALDH1A1CHEK2CNR1PDE7BPRMT5
SCHEMBL8515983 0.81 CHEK2 (0.40) ALDH1A1CHEK2PDE7BPRMT5TRPV1
SCHEMBL5772427 0.78 F2 (0.38) CHEK1
SCHEMBL5769284 0.78 CHEK2 (0.40) ALDH1A1CHEK2PDE7BPRMT5TRPV1
SCHEMBL5773134 0.75 ATM (0.39) ALDH1A1CHEK2PDE7BPRMT5TRPV1
SCHEMBL8516353 0.72 F2 (0.40) CCNT1CDK2
SCHEMBL5769599 0.72 ATM (0.38) ALDH1A1CHEK2PDE7BPRMT5TRPV1
SCHEMBL8519327 0.70 PIK3CA (0.39) ALDH1A1CNR1FGFR1
SCHEMBL5769605 0.68 TRPV1 (0.37) ALDH1A1CHEK2PDE7BPRMT5TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066899-A1 NOVEL THROMBIN INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) AG (CH) 2006-06-29 WO disclosed
EP-1674464-A1 Novel thrombin inhibitors Santhera Pharmaceuticals (Schweiz) GmbH (CH) 2006-06-28 EP disclosed
EP-1674464-A1 Novel thrombin inhibitors Santhera Pharmaceuticals (Schweiz) GmbH (CH) 2006-06-28 EP disclosed