SCHEMBL5772031

SCHEMBL5772031

Nc1nc2ccc(-c3nc[nH]c3-c3ccccc3)cc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.59
CYP3A4 P08684 2/20 0.54
KDM4E B2RXH2 2/20 0.54
MAPT P10636 2/20 0.54
IDO1 P14902 4/20 0.53
ABL1 P00519 1/20 0.45
FABP6 P51161 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MASP2 O00187 1/20 0.44
MEN1 O00255 1/20 0.44
NUDT1 P36639 1/20 0.44
KMT2A Q03164 1/20 0.44
AOC3 Q16853 1/20 0.44
PLAU P00749 1/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
BACE1 P56817 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18041623 0.95 CYP3A4 (0.54) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL5772038 0.90 CYP3A4 (0.54) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL11712219 0.80 ALDH1A1 (0.58) MAPK14CYP3A4KDM4EMAPTABL1
SCHEMBL4834100 0.76 MAPT (0.44) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL4840197 0.75 MAPK14 (0.65) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL4839601 0.74 MAPK14 (1.00) MAPK14CYP3A4
SCHEMBL224770 0.73 KDM4E (1.00) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL18041756 0.72 RAB9A (0.57) MAPK14CYP3A4KDM4EMAPTIDO1
SCHEMBL26003342 0.72 IDO1 (0.63) MAPK14CYP3A4KDM4EMAPTIDO1
Bromide SCHEMBL31020961 0.71 KDM4E (0.96) MAPK14CYP3A4KDM4EMAPTIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-B1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE LILLY CO ELI (US) 2006-10-25 EP disclosed