SCHEMBL5772297

SCHEMBL5772297

CCOC(=O)C(C(=O)Nc1c(OC)cc(OC)cc1OC)c1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 1/20 0.58
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5797214 0.86 MEN1 (0.51)
SCHEMBL7506148 0.81 MEN1 (0.46)
SCHEMBL27554209 0.80 MMP8 (0.50) MMP8CA12CA1CA2CA9
SCHEMBL7189265 0.79 MMP8 (0.49) MMP8CA12CA1CA2CA9
SCHEMBL9435341 0.76 MMP8 (0.62) MMP8CA12CA1CA2CA9
SCHEMBL28474562 0.75 MMP8 (0.73) MMP8CA12CA1CA2CA9
SCHEMBL7052592 0.75 MEN1 (0.48)
SCHEMBL15944495 0.74 MMP8 (0.77) MMP8CA12CA1CA2CA9
Ethyl Acetate SCHEMBL8909263 0.74 SMN1; SMN2 (0.53)
SCHEMBL266419 0.73 MMP8 (0.74) MMP8CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203767-B1 Heterocyclic-substituted alkylamide acat inhibitors WARNER LAMBERT CO (US) 2006-01-04 EP disclosed
EP-1203767-A1 Heterocyclic-substituted alkylamide acat inhibitors WARNER-LAMBERT COMPANY (US) 2002-05-08 EP disclosed
EP-0684945-A1 HETEROCYCLIC-SUBSTITUTED ALKYL AMIDE ACAT INHIBITORS WARNER-LAMBERT COMPANY (US) 1995-12-06 EP disclosed
US-5441975-A Anticholesterol agent WARNER-LAMBERT COMPANY (US) 1995-08-15 US disclosed
US-5366987-A Enzyme inhibitors, anticholesterol WARNER-LAMBERT COMPANY (US) 1994-11-22 US disclosed
WO-1994019330-A1 HETEROCYCLIC-SUBSTITUTED ALKYL AMIDE ACAT INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-09-01 WO disclosed