SCHEMBL5772672

SCHEMBL5772672

Cn1c2ccccc2c(=O)c2c(O)c(OCCN3CCCCC3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.50
HTR2C P28335 4/20 0.50
HTR2B P41595 4/20 0.50
KDM1A O60341 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD3 P35462 1/20 0.44
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ABCB1 P08183 1/20 0.43
OPRK1 P41145 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777884 0.97 KDM1A (0.48) HTR2AHTR2CHTR2BKDM1AMAPT
SCHEMBL5770520 0.91 KDM1A (0.47) HTR2AHTR2CHTR2BKDM1AMAPT
SCHEMBL5749161 0.86 TDP1 (0.51) HTR2AHTR2CHTR2BMAPTHTT
SCHEMBL5747101 0.85 TDP1 (0.52) HTR2AHTR2CHTR2BMAPTHTT
SCHEMBL5776994 0.83 HTT (0.52) KDM1AMAPTHTTMEN1GAA
SCHEMBL5773781 0.81 HTT (0.50) KDM1AMAPTHTTMEN1GAA
SCHEMBL5774116 0.81 HRH3 (0.53) HTR2AMAPTMEN1KMT2ATDP1
SCHEMBL5772233 0.80 KDM1A (0.49) KDM1AMAPTHTTGAAKMT2A
SCHEMBL5775529 0.80 KDM1A (0.49) KDM1AMAPTHTTGAAKMT2A
SCHEMBL5772950 0.79 G6PD (0.49) KDM1AMAPTHTTGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed