SCHEMBL5770520

SCHEMBL5770520

Cn1c2ccccc2c(=O)c2c(O)c(OCCCN3CCC3)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.47
MAPT P10636 2/20 0.47
HTT P42858 1/20 0.47
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
CHEK1 O14757 1/20 0.43
CDK1 P06493 1/20 0.43
WEE1 P30291 1/20 0.43
HTR5A P47898 2/20 0.43
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
RAD52 P43351 1/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777884 0.94 KDM1A (0.48) KDM1AMAPTHTTCYP2D6CYP2C19
SCHEMBL5772672 0.91 HTR2A (0.50) KDM1AMAPTHTTCYP2D6CYP2C19
SCHEMBL5745434 0.86 CYP2D6 (0.50) MAPTHTTCYP2D6CYP2C19L3MBTL1
SCHEMBL5774116 0.83 HRH3 (0.53) MAPTCYP2D6CYP2C19L3MBTL1KMT2A
SCHEMBL5776994 0.83 HTT (0.52) KDM1AMAPTHTTCYP2C19L3MBTL1
SCHEMBL5775529 0.82 KDM1A (0.49) KDM1AMAPTHTTCYP2C19LMNA
SCHEMBL5770337 0.81 KDM1A (0.48) KDM1AMAPTHTTCYP2C19LMNA
SCHEMBL5773781 0.81 HTT (0.50) KDM1AMAPTHTTCYP2C19CHEK1
SCHEMBL5822008 0.80 G6PD (0.48) KDM1AMAPTHTTCYP2C19HPGD
SCHEMBL5772233 0.80 KDM1A (0.49) KDM1AMAPTHTTCYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed