SCHEMBL5773768

SCHEMBL5773768

CC(C)(C)OC(=O)Nc1ccc2c(c1)Cc1cccc(Br)c1S2.CC(C)(C)OC(=O)OC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.39
NR1I3 Q14994 5/20 0.38
HDAC3 O15379 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC8 Q9BY41 4/20 0.36
HDAC10 Q969S8 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
CYP17A1 P05093 1/20 0.35
CA1 P00915 2/20 0.35
DRD2 P14416 1/20 0.35
CA2 P00918 1/20 0.35
LIPE Q05469 1/20 0.35
CYP1A2 P05177 1/20 0.34
ADRA2A P08913 1/20 0.34
MAOA P21397 1/20 0.34
SLC6A2 P23975 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3173494 0.95 ATM (0.40) ATMNR1I3HDAC3HDAC1HDAC2
SCHEMBL2762684 0.83 ATM (0.41) ATMNR1I3HDAC3HDAC1HDAC2
SCHEMBL27645340 0.79 ATM (0.42) ATMCA1CA2CYP1A2ADRA2A
SCHEMBL2763052 0.78 MMP8 (0.38) ATMNR1I3MMP3MMP8
SCHEMBL3167857 0.77 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC8HDAC10
SCHEMBL13376023 0.76 MMP8 (0.38) ATMNR1I3DRD2MMP3MMP8
SCHEMBL3165587 0.76 ATM (0.38) ATMNR1I3PRMT5WDR77CYP17A1
SCHEMBL17827825 0.72 SIRT2 (0.40) NR1I3HDAC3HDAC1HDAC2HDAC8
SCHEMBL17827852 0.70 NR1I3 (0.41) NR1I3HDAC3HDAC1HDAC2HDAC8
SCHEMBL1114945 0.69 RAB9A (0.56) NR1I3CYP17A1CA1CYP1A2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654257-A1 AMINOPYRONES AND THEIR USE AS ATM INHIBITORS Kudos Pharmaceuticals Limited (GB) 2006-05-10 EP disclosed
WO-2005016919-A1 AMINOPYRONES AND THEIR USE AS ATM INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2005-02-24 WO disclosed