SCHEMBL5774466

SCHEMBL5774466

CCOC(=O)Oc1[nH]c2cc(Cl)cc(Cl)c2c1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.46
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
BLM P54132 2/20 0.39
KMT2A Q03164 2/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KRAS P01116 1/20 0.39
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9573782 0.84 GRIN2D (0.43) ALOX15MEN1CYP1A2BLMKMT2A
SCHEMBL9573817 0.81 CA12 (0.38) ALOX15MEN1CYP1A2BLMKMT2A
SCHEMBL5777941 0.80 POLB (0.40) ALOX15MEN1CYP1A2KMT2AGRIN2D
SCHEMBL5397544 0.80 ALOX15 (0.66) ALOX15CYP1A2HPGDCYP2C19
SCHEMBL5812465 0.78 ALOX15 (0.54) ALOX15MEN1CYP1A2KMT2AHPGD
SCHEMBL7255962 0.77 MEN1 (0.42) ALOX15MEN1CYP1A2BLMKMT2A
SCHEMBL4337035 0.76 GRIN1 (0.48) ALOX15MEN1KMT2ACYP2C9HPGD
SCHEMBL5776615 0.74 KDM4E (0.45) ALOX15MEN1KMT2AHPGDTSHR
SCHEMBL4344101 0.74 GRIN1 (0.39) MEN1CYP1A2BLMKMT2AHPGD
SCHEMBL5775281 0.72 KDM4E (0.48) ALOX15MEN1KMT2AHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472221-B1 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN GRUENENTHAL GMBH (DE) 2006-03-22 EP disclosed
EP-1472221-A2 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN Grünenthal GmbH (DE) 2004-11-03 EP disclosed
WO-2003037863-A2 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN Grünenthal GmbH (DE) 2003-05-08 WO disclosed
WO-1994013637-A1 HYDROXYIMINOALKYLINDOLE CARBOXYLIC ACID DERIVATIVES USED AS ANTAGONISTS OF EXCITATORY AMINO ACIDS BASF AKTIENGESELLSCHAFT (DE) 1994-06-23 WO disclosed