SCHEMBL5812465

SCHEMBL5812465

CCOC(=O)Oc1[nH]c2ccc(Cl)cc2c1C=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 5/20 0.54
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.46
CYP1A2 P05177 1/20 0.46
XBP1 P17861 1/20 0.46
CYP2C19 P33261 1/20 0.46
CSF1R P07333 1/20 0.44
LMNA P02545 3/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALOX5 P09917 2/20 0.42
SIRT1 Q96EB6 3/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5775281 0.88 KDM4E (0.48) ALOX15ALDH1A1HPGDLMNAMAPT
SCHEMBL9240047 0.85 ALDH1A1 (0.50) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL9573776 0.84 ALDH1A1 (0.49) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL9242488 0.82 ALDH1A1 (0.48) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL5776615 0.82 KDM4E (0.45) ALOX15ALDH1A1HPGDLMNAMAPT
SCHEMBL9573800 0.81 TUBB4A (0.51) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL1503856 0.80 ALOX15 (0.81) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL29954955 0.80 ALOX15 (0.81) ALOX15ALDH1A1HPGDCYP1A2XBP1
SCHEMBL5774466 0.78 ALOX15 (0.46) ALOX15HPGDCYP1A2CYP2C19LMNA
SCHEMBL9573804 0.76 ALOX15 (0.52) ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472221-B1 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN GRUENENTHAL GMBH (DE) 2006-03-22 EP disclosed
EP-1472221-A2 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN Grünenthal GmbH (DE) 2004-11-03 EP disclosed
WO-2003037863-A2 SUBSTITUTED INDOLES, METHOD FOR PRODUCTION AND USE THEREOF FOR THE INHIBITION OF PAIN Grünenthal GmbH (DE) 2003-05-08 WO disclosed