SCHEMBL5775682

SCHEMBL5775682

O=C(O)Oc1nc(-c2ccccc2)ncc1NC(=O)OCc1cc2cc(-c3ccc(F)cc3)ccc2o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 4/20 0.41
MAOB P27338 3/20 0.38
HDAC3 O15379 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
ADCY8 P40145 2/20 0.34
ADCY1 Q08828 2/20 0.34
ELANE P08246 1/20 0.33
ASAH1 Q13510 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5776630 0.96 MAOB (0.40) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL5775678 0.88 MGLL (0.43) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL5778231 0.88 MAOB (0.36) MAOBHDAC3HDAC1HDAC2CYP1A2
SCHEMBL6167634 0.83 MGLL (0.46) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL5777269 0.83 MAOB (0.41) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL6166144 0.83 MGLL (0.46) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL5774430 0.81 MAOB (0.40) MGLLMAOBMAPTLMNAFFAR1
SCHEMBL6164514 0.80 MGLL (0.48) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL6166379 0.80 MGLL (0.48) MGLLMAOBHDAC3HDAC1HDAC2
SCHEMBL6165379 0.80 MGLL (0.41) MGLLMAOBHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368345-B1 ALKOXYCARBONYLAMINO HETEROARYL CARBOXYLIC ACID DERIVATIVES AS IP ANTAGONISTS HOFFMANN LA ROCHE (CH) 2006-03-22 EP claimed