SCHEMBL5775765

SCHEMBL5775765

NC(=S)CCc1cccc(NC(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.53
ITGA2B P08514 1/20 0.53
MAPT P10636 5/20 0.53
GAA P10253 2/20 0.53
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
RECQL P46063 1/20 0.50
GFER P55789 1/20 0.49
SIRT1 Q96EB6 1/20 0.48
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
LMNA P02545 1/20 0.47
ALOX12 P18054 1/20 0.47
HTT P42858 1/20 0.45
SELL P14151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777508 0.88 ITGB3 (0.56) ITGB3ITGA2BMAPTGAAMEN1
SCHEMBL4752320 0.81 HTR6 (0.55) ITGB3ITGA2BMAPTGAAGFER
SCHEMBL4337810 0.79 TRPV1 (0.53) ITGB3ITGA2BMAPTGAAALDH1A1
SCHEMBL4334746 0.78 MAOA (0.58) ITGB3ITGA2BMAPTGAAALDH1A1
SCHEMBL16246034 0.78 MAPT (0.54) ITGB3ITGA2BMAPTGAAMEN1
SCHEMBL13735094 0.78 MAPT (0.50) ITGB3ITGA2BMAPTGAAMEN1
SCHEMBL3003205 0.77 CFD (0.59) MAPTGAACYP1A2CYP2C9CYP2C19
SCHEMBL8059186 0.76 KMT2A (0.55) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL1074012 0.75 MAPT (0.68) MAPTGAAALDH1A1GFERRAB9A
SCHEMBL4523190 0.75 SIRT2 (0.60) ITGB3ITGA2BMAPTGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed