SCHEMBL5776842

SCHEMBL5776842

Clc1ccccc1-c1[c]ccc(Cl)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 3/20 0.36
LMNA P02545 2/20 0.36
DPP4 P27487 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HSD11B1 P28845 1/20 0.34
NOTUM Q6P988 3/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IDO1 P14902 1/20 0.33
PTPRC P08575 1/20 0.32
LDHA P00338 1/20 0.32
P2RX7 Q99572 1/20 0.32
GALR1 P47211 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520665 0.82 CYP1A2 (0.34) ALDH1A1HSD11B1NOTUMIDO1
SCHEMBL3990580 0.78 CYP2A6 (0.44) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL6576709 0.77 CYP2A6 (0.38) CYP2A6NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL8560761 0.77 CYP2A6 (0.43) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL9988583 0.72 ALDH1A1 (0.46) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL10506626 0.72 PLA2G7 (0.41) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL7458982 0.72 CYP2A6 (0.59) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL9512604 0.71 CYP2A6 (0.41) CYP2A6NPC1RAB9ASMN1; SMN2TP53
SCHEMBL4313272 0.71 NOTUM (0.39) CYP2A6TSHRNOTUMIDO1P2RX7
SCHEMBL9729126 0.71 CYP2A6 (0.41) CYP2A6NPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615890-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY (US) 2006-01-18 EP disclosed
WO-2004089903-A1 PIPERIDINE DERIVATIVES AS RENIN INHIBITORS FOR THE TREATMENT OF HYPERTENSION WARNER-LAMBERT COMPANY LLC (US) 2004-10-21 WO disclosed