SCHEMBL5777302

SCHEMBL5777302

Fc1cc(Sc2ccc(Cl)cc2)c2c(Sc3ccc(Cl)cc3)c3n(c2c1F)CC[CH]3

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 6/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR1A P08908 3/20 0.31
HTR3A P46098 3/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 2/20 0.31
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777307 0.78 TBXA2R (0.32) TBXA2RPTGDR2MEN1KMT2AHTR1A
SCHEMBL5773536 0.72 TBXA2R (0.56) TBXA2RPTGDR2HTR1AAKR1B1
SCHEMBL5778173 0.68 TBXA2R (0.50) TBXA2RPTGDR2AKR1B1
SCHEMBL5776538 0.66 TBXA2R (0.39) TBXA2RPTGDR2AKR1B1
SCHEMBL21984840 0.57 MEN1 (0.46) MEN1KMT2AHTR1AHTR3ACYP1A2
SCHEMBL3546610 0.55 MEN1 (0.47) PTGDR2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL3541411 0.55 MEN1 (0.47) TBXA2RPTGDR2MEN1KMT2ACYP1A2
SCHEMBL9476350 0.53 MAOA (0.64) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL481976 0.53 MAOA (0.64) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9475224 0.53 MAOA (0.64) MEN1KMT2ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed